Ozmosi | Varlitinib Drug Profile
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Varlitinib

Alternative Names: varlitinib, arry-334543, aslan-001, aslan001, aslan 001
Clinical Status: Inactive
Latest Update: 2025-09-10
Latest Update Note: Clinical Trial Update

Product Description

Mechanisms of Action: TK Inhibitor, HER2 Inhibitor, EGFR Inhibitor

Novel Mechanism: No

Modality: Small Molecule

Route of Administration: Oral

FDA Designation: *

Approval Status: Not Approved

Approved Countries: None

Approved Indications: None

Known Adverse Events: None

Company: Aslan
Company Location: SINGAPORE U0 239920
Company CEO:
Additional Commercial Interests: None

Clinical Description

Countries in Clinic:

Active Clinical Trial Count:

Recent & Upcoming Milestones

Highest Development Phases

Phase 3: Papillary Carcinoma|Cholangiocarcinoma|Gallbladder Cancer|Biliary Tract Cancer|Gastrointestinal Cancer

Phase 2: Breast Cancer|Biliary Tract Cancer|Pancreatic Cancer|Hepatocellular Carcinoma|Cholangiocarcinoma|Gastrointestinal Cancer

Phase 1: Oncology Solid Tumor Unspecified|Gallbladder Cancer|Breast Cancer|Biliary Tract Cancer|Papillary Carcinoma|Cholangiocarcinoma|Healthy Volunteers

Trial ID

Trial

Phase

Trial Status

Disease

Primary Completion Date

Probability of Success

Latest Trial Update Date

Data Updated

ACTRN12619001528145p

2006-7041-83/hah

N/A

Not yet recruiting

Obesity|Weight Gain

2020-07-31

NCT02435927

ASLAN001-002SG

P1

Unknown status

Oncology Solid Tumor Unspecified

2021-06-01

2023-04-15

Primary Endpoints

NCT03082053

ASLAN001-010

P1

Completed

Biliary Tract Cancer

2017-12-07

2025-08-27

Primary Endpoints|Treatments

NCT03368846

ASLAN001-018

P1

Completed

Healthy Volunteers

2017-12-06

2023-04-15

Primary Endpoints|Treatments

NCT02648425

ASLAN001-002

P1

Completed

Oncology Solid Tumor Unspecified

2017-06-12

2023-04-15

NCT00637702

ARRAY-543-103

P1

Completed

Oncology Solid Tumor Unspecified

2012-10-01

2020-10-07

Primary Endpoints|Treatments

NCT00710736

ARRAY-543-204

P1

Completed

Oncology Solid Tumor Unspecified

2011-04-01

2020-10-07

NCT00833326

ARRAY-543-104

P1

Completed

Oncology Solid Tumor Unspecified

2010-07-01

2020-10-07

Primary Endpoints|Treatments

NCT00278902

ARRY-0501

P1

Completed

Breast Cancer

2009-06-01

2020-10-16

JapicCTI-173497

JapicCTI-173497

P1

Completed

Gallbladder Cancer|Biliary Tract Cancer|Papillary Carcinoma|Cholangiocarcinoma

None

NCT02992340

ASLAN001-007

P2

Terminated

Biliary Tract Cancer

2020-06-16

2023-04-15

NCT03129074

ASLAN001-016

P2

Withdrawn

Biliary Tract Cancer

2020-03-01

2023-04-15

Primary Endpoints|Treatments

NCT07166367

ASLAN001-006

P2

Terminated

Breast Cancer

2020-01-14

2025-09-11

Primary Endpoints|Treatments

NCT03231176

ASLAN001-008

P2

Completed

Biliary Tract Cancer

2019-07-05

2023-04-15

Primary Endpoints|Treatments

NCT03499626

HC01/12/16

P2

Unknown status

Hepatocellular Carcinoma

2019-05-05

2021-05-07

Primary Endpoints|Treatments|Trial Status

NCT02396108

NCT02396108

P2

Unknown status

Breast Cancer

2018-03-01

2019-03-20

Treatments

NCT02609958

ASLAN001-005

P2

Completed

Cholangiocarcinoma

2017-07-07

2023-04-15

Primary Endpoints|Treatments

NCT02338245

ASLAN001-003

P2

Completed

Breast Cancer

2016-05-19

2023-04-15

Primary Endpoints|Treatments

NCT01614522

ASLAN001-001

P2

Completed

Gastrointestinal Cancer

2013-03-01

2023-04-15

Primary Endpoints|Treatments

NCT00862524

ARRAY-543-206

P2

Completed

Pancreatic Cancer

2011-02-01

2019-03-18

JapicCTI-183951

JapicCTI-183951

P3

Unknown

Papillary Carcinoma|Gallbladder Cancer|Cholangiocarcinoma|Biliary Tract Cancer

2019-12-31

NCT03093870

TreeTopp

P3

Completed

Biliary Tract Cancer

2019-11-12

28%

2023-04-15

Primary Endpoints|Treatments

2017-000114-30

TreeTopp

P3

Terminated

Biliary Tract Cancer

2019-11-12

2022-03-13

Treatments

2017-001833-15

2017-001833-15

P3

Terminated

Gastrointestinal Cancer

2019-01-31

2025-06-28

Treatments

NCT03130790

First Line

P3

Completed

Gastrointestinal Cancer

2018-12-20

2023-04-15

Primary Endpoints|Treatments