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Timapiprant

Alternative Names: timapiprant, oc000459, oc-459, oc459, oc 459, oc-000459
Latest Update: 2023-10-30
Latest Update Note: Clinical Trial Update

Product Description

OC000459, a potent, selective, and orally active D prostanoid receptor 2 antagonist that inhibits mast cell-dependent activation of T helper 2 lymphocytes and eosinophils

Mechanisms of Action: CRTH2 Antagonist

Novel Mechanism: Yes

Modality: Small Molecule

Route of Administration: Oral

FDA Designation: None *

Approval Status: Not Approved

Approved Countries: None

Approved Indications: None

Known Adverse Events: None

Company: Oxagen
Company Location:
Company CEO:
Additonal Commercial Interests: None

Clinical Description

Map of Global Clinical Trials for Timapiprant

Countries in Clinic:

Active Clinical Trial Count: 1

Highest Development Phases

Phase 3: Asthma

Trial

Phase

Trial Status

Disease

Primary Completion Date

Probability of Success

2018-003548-22

P3

Completed

Asthma

2021-02-01

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