Ozmosi | BMB-201 Drug Profile
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BMB-201

Alternative Names: BMB-201, BMB201, BMB 201
Clinical Status: Active
Latest Update: 2025-09-04
Latest Update Note: News Article

Product Description

BMB-201, a selective 5-HT2A/2C receptor agonist, was designed to harness the analgesic potential of serotonin modulation without the hallucinogenic effects commonly associated with 5-HT2A activation. As a prodrug of BMB-A39a, it exhibits minimal activity at the 5-HT2B receptor, ensuring a reduced risk of side effects. (Sourced from: https://brightmindsbio.com/bright-minds-biosciences-proprietary-compound-bmb-201-5-ht2c-2a-mixed-agonist-demonstrated-similar-efficacy-to-morphine-in-preclinical-pain-models/)

Mechanisms of Action: 5-HT2C Agonist

Novel Mechanism: No

Modality: Small Molecule

Route of Administration: N/A

FDA Designation: *

Approval Status: Not Approved

Approved Countries: None

Approved Indications: None

Known Adverse Events: None

Company: Bright Minds Biosciences
Company Location: Eastern America
Company CEO:
Additional Commercial Interests: None

Clinical Description

Countries in Clinic:

Active Clinical Trial Count:

Recent & Upcoming Milestones

  • Clinical Outcomes Reported - Bright Minds Biosciences presented P0 Pain Unspecified results on 2024-10-16 for BMB-201

Highest Development Phases

Phase 0: Pain Unspecified

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