Ozmosi | Lobeline Drug Profile
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Lobeline

Alternative Names: lobeline
Clinical Status: Inactive
Latest Update: 2025-06-18
Latest Update Note: News Article

Product Description

Mechanisms of Action: VMAT1 Inhibitor, NIACR Antagonist

Novel Mechanism: Yes

Modality: Small Molecule

Route of Administration: Oral, Sublingual

FDA Designation: *

Approval Status: Not Approved

Approved Countries: China | Taiwan

Approved Indications: None

Known Adverse Events: None

Company: Yaupon
Company Location:
Company CEO:
Additional Commercial Interests: None

Clinical Description

Countries in Clinic:

Active Clinical Trial Count:

Recent & Upcoming Milestones

Highest Development Phases

Phase 2: Attention Deficit Disorder with Hyperactivity

Phase 1: Amphetamine-Related Disorders|Methamphetamine Dependence

Trial ID

Trial

Phase

Trial Status

Disease

Primary Completion Date

Probability of Success

Latest Trial Update Date

Data Updated

NCT00100074

NIDA-CPU-0007-1

P1

Unknown status

Amphetamine-Related Disorders

None

2019-03-21

Treatments

NCT00439504

NIDA-CPU-0012-1

P1

Unknown status

Amphetamine-Related Disorders|Methamphetamine Dependence

None

2019-03-21

Treatments

NCT00519259

NIDA-CPU-0009-1

P1

Unknown status

Methamphetamine Dependence|Amphetamine-Related Disorders

None

2019-03-21

Treatments

NCT00664703

R43MH081553

P2

Completed

Attention Deficit Disorder with Hyperactivity

2010-01-01

2019-03-18