Ozmosi | BGB-53038 Drug Profile
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BGB-53038

Alternative Names: BGB-53038, BGB 53038, BGB53038
Clinical Status: Active
Latest Update: 2025-07-10
Latest Update Note: Clinical Trial Update

Product Description

PanKRAS inhibitor 2G for lung and GI cancers in preclinical development. (Sourced from: https://www.beigene.com/science/pipeline/)

Mechanisms of Action: KRAS Inhibitor

Novel Mechanism: Yes

Modality: Unknown

Route of Administration: Oral

FDA Designation: *

Approval Status: Not Approved

Approved Countries: None

Approved Indications: None

Known Adverse Events: None

Company: BeiGene
Company Location:
Company CEO: John V. Oyler
Additional Commercial Interests: None

Clinical Description

Map of Global Clinical Trials for BGB-53038

Countries in Clinic: Australia, China, Korea, New Zealand, South Korea, Spain, United States

Active Clinical Trial Count: 2

Recent & Upcoming Milestones

Highest Development Phases

Phase 1: Adenocarcinoma|Colorectal Cancer|Esophageal Cancer|Gastrointestinal Cancer|Non-Small-Cell Lung Cancer|Oncology Solid Tumor Unspecified|Pancreatic Cancer|Pancreatic Ductal Carcinoma|Squamous Cell Carcinoma

Trial ID

Trial

Phase

Trial Status

Disease

Primary Completion Date

Probability of Success

Latest Trial Update Date

Data Updated

NCT06585488

BGB-53038-101

P1

Recruiting

Gastrointestinal Cancer|Pancreatic Ductal Carcinoma|Pancreatic Cancer|Adenocarcinoma|Non-Small-Cell Lung Cancer|Colorectal Cancer|Esophageal Cancer|Squamous Cell Carcinoma

2026-12-01

12%

2025-07-11

CTR20250063

CTR20250063

P1

Recruiting

Oncology Solid Tumor Unspecified

None

2025-10-05

Patient Enrollment|Treatments