Ozmosi | Azasetron Drug Profile
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Azasetron

Pronounced as: ay-ZA-se-tron

Alternative Names: azasetron
Clinical Status: Active
Latest Update: 2026-07-02
Latest Update Note: Clinical Trial Update

Product Description

Azasetron (Serotone) is a potent and selective 5-HT3 receptor antagonist, and classified as benzamide derivative. It has a different chemical structure from indole-type 5-HT3 receptor antagonists such as granisetron, ondansetron, ramosetron and tropisetron. (Sourced from: https://pubmed.ncbi.nlm.nih.gov/10396331/)

Mechanisms of Action: 5-HT3 Antagonist

Novel Mechanism: No

Modality: Small Molecule

Route of Administration: N/A

FDA Designation: *

Approval Status: Not Approved

Approved Countries: None

Approved Indications: None

Company: Sensorion
Company Location:
Company Founding Year: None
Additional Commercial Interests: None

Clinical Description

Map of Global Clinical Trials for Azasetron

Countries in Clinic: France

Active Clinical Trial Count: 2

Recent & Upcoming Milestones

Highest Development Phases

Phase 2: Hearing Loss

Trial ID

Trial

Phase

Trial Status

Disease

Primary Completion Date

Probability of Success

Latest Trial Update Date

Data Updated

NCT05628233

NOTOXIS

P2

Completed

Hearing Loss

2025-04-16

2026-07-03

Primary Endpoints

2024-511713-38-00

SENS-401-202

P2

Recruiting

Hearing Loss

2025-03-31

2025-05-02

Treatments