Ozmosi | Orantinib Drug Profile
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Orantinib

Alternative Names: orantinib, tsu-68
Clinical Status: Inactive
Latest Update: 2023-06-08
Latest Update Note: PubMed Publication

Product Description

Mechanisms of Action: FGFR Antagonist, PGFR Inhibitor, VEGFR Inhibitor, TK Inhibitor

Novel Mechanism: No

Modality: Small Molecule

Route of Administration: Oral

FDA Designation: *

Approval Status: Not Approved

Approved Countries: None

Approved Indications: None

Known Adverse Events: None

Company: Taiko Co
Company Location: Asia Pacific
Company CEO:
Additional Commercial Interests: None

Clinical Description

Countries in Clinic:

Active Clinical Trial Count:

Recent & Upcoming Milestones

Highest Development Phases

Phase 3: Hepatocellular Carcinoma

Phase 2: Hepatocellular Carcinoma|Breast Cancer|Gastrointestinal Cancer|Colorectal Cancer

Phase 1: Breast Cancer|Pancreatic Cancer|Plasmacytoma|Lung Cancer|Hepatocellular Carcinoma|Non-Small-Cell Lung Cancer|Prostate Cancer|Multiple Myeloma|Kidney Cancer|Colorectal Cancer|Gastrointestinal Cancer|Oncology Solid Tumor Unspecified

Trial ID

Trial

Phase

Trial Status

Disease

Primary Completion Date

Probability of Success

Latest Trial Update Date

Data Updated

JapicCTI-121970

JapicCTI-121970

P1

Completed

Hepatocellular Carcinoma

2013-03-31

JapicCTI-101323

JapicCTI-101323

P1

Completed

Non-Small-Cell Lung Cancer

2012-03-31

JapicCTI-111402

JapicCTI-111402

P1

Completed

Colorectal Cancer

2010-05-31

NCT00024206

NCI-2012-02412

P1

Completed

Oncology Solid Tumor Unspecified

2003-07-01

2020-10-26

Primary Endpoints|Treatments

NCT00024063

CDR0000068888

P1

Unknown status

Breast Cancer|Pancreatic Cancer|Plasmacytoma|Lung Cancer|Prostate Cancer|Multiple Myeloma|Kidney Cancer|Colorectal Cancer|Gastrointestinal Cancer

None

2019-03-21

JapicCTI-111403

JapicCTI-111403

P2

Completed

Colorectal Cancer

2012-12-31

JapicCTI-101327

JapicCTI-101327

P2

Completed

Gastrointestinal Cancer

2012-03-31

JapicCTI-101178

JapicCTI-101178

P2

Completed

Breast Cancer

2011-03-31

JapicCTI-111404

JapicCTI-111404

P2

Completed

Breast Cancer

2011-01-04

JapicCTI-101087

JapicCTI-101087

P2

Completed

Hepatocellular Carcinoma

2010-12-31

NCT00784290

Taiho132070

P2

Completed

Hepatocellular Carcinoma

2010-10-01

2019-03-18

Treatments

JapicCTI-101354

JapicCTI-101354

P3

Terminated

Hepatocellular Carcinoma

2016-05-31

NCT01465464

ORIENTAL

P3

Terminated

Hepatocellular Carcinoma

2014-06-01

2019-03-19

Treatments