Ozmosi | Mepyramine Drug Profile
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Mepyramine

Alternative Names: mepyramine
Clinical Status: Inactive
Latest Update: 2025-04-30
Latest Update Note: Clinical Trial Update

Product Description

Mepyramine, a histamine H1 receptor inverse agonist, binds preferentially to a G protein-coupled form of the receptor and sequesters G protein (Sourced from: https://pubmed.ncbi.nlm.nih.gov/15192105/)

Mechanisms of Action: H1 Inverse Agonist

Novel Mechanism: No

Modality: Small Molecule

Route of Administration: Topical

FDA Designation: *

Approval Status: Approved

Approved Countries: Algeria | Bangladesh | Dominican Republic | Ecuador | France | Hong Kong | India | Indonesia | Ireland | Lebanon | Malta | Mexico | New Zealand | Pakistan | Peru | Portugal | South Africa | Spain | Taiwan | Turkey | United Kingdom | Uruguay

Approved Indications: None

Known Adverse Events: None

Company: None
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Additional Commercial Interests: None

Clinical Description

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